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Pierre Roubert

Observed names: P Roubert, P. Roubert
Institution: Ipsen (France)
OpenAlex ID: A5109034433
Analysis of the therapeutic functions of novel melanocortin receptor agonists in MC3R- and MC4R-deficient C57BL/6J mice
2009 · K. Ganesh Kumar, Gregory M. Sutton, et al. · Peptides · 96
Regulation of atrial natriuretic factor receptors by angiotensin II in rat vascular smooth muscle cells.
1988 · P E Chabrier, P Roubert, et al. · Journal of Biological Chemistry · 73
Anticancer Activity of BIM-46174, a New Inhibitor of the Heterotrimeric Gα/Gβγ Protein Complex
2006 · Grégoire P. Prévost, Marie O. Lonchampt, et al. · Cancer Research · 62
Identification of Potent Non-Peptide Somatostatin Antagonists with sst3 Selectivity
2001 · Lydie Poitout, Pierre Roubert, et al. · Journal of Medicinal Chemistry · 61
Angiotensin II and phorbol-esters potently down-regulate endothelin (ET-1) binding sites in vascular smooth muscle cells
1989 · Pierre Roubert, Véronique Gillard, et al. · Biochemical and Biophysical Research Communications · 56
Vascular Mechanism of Action of Endothelin-1
1989 · Pierre étienne Chabrier, Michel Auguet, et al. · Journal of Cardiovascular Pharmacology · 53
Down-regulation of atrial natriuretic factor receptors and correlation with cGMP stimulation in rat cultured vascular smooth muscle cells
1987 · P. Roubert, M.O. Lonchampt, et al. · Biochemical and Biophysical Research Communications · 52
3-Thio-1,2,4-triazoles, novel somatostatin sst2/sst5 agonists
2005 · Marie-Odile Contour-Galcéra, Alban Sidhu, et al. · Bioorganic & Medicinal Chemistry Letters · 49
Specific binding of atrial natriuretic factor in brain microvessels.
1987 · P E Chabrier, P Roubert, et al. · Proceedings of the National Academy of Sciences · 49
Novel pharmacological MC4R agonists can efficiently activate mutated MC4R from obese patient with impaired endogenous agonist response
2010 · Pierre Roubert, Béatrice Dubern, et al. · Journal of Endocrinology · 40
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Identification of a novel series of benzimidazoles as potent and selective antagonists of the human melanocortin-4 receptor
2007 · Lydie Poitout, Valérie Brault, et al. · Bioorganic & Medicinal Chemistry Letters · 34
Endothelin receptor subtypes A and B are up-regulated in an experimental model of acute renal failure.
1994 · P Roubert, V Gillard-Roubert, et al. · Molecular Pharmacology · 30
Comparison of the Bronchopulmonary and Pressor Activities of Endothelin Isoforms ET-1, ET-2, and ET-3 and Characterization of Their Binding Sites in Guinea Pig Lung
1991 · Francoise Pons, Isabelle Loquet, et al. · American Review of Respiratory Disease · 29
Effects and specific binding sites of endothelin in human lung preparations
1991 · C. Brink, V. Gillard, et al. · Pulmonary Pharmacology · 29
Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5
2001 · Marie-Odile Contour-Galcéra, Lydie Poitout, et al. · Bioorganic & Medicinal Chemistry Letters · 22
Down-regulation of Endothelin Binding Sites in Rat Vascular Smooth Muscle Cells
1990 · P. Roubert, V. Gillard, et al. · American Journal of Hypertension · 22
Somatostatin-14 Mainly Binds the Somatostatin Receptor Subtype 2 in Human Neuroblastoma Tumors
2008 · Grégoire Prévost, Nathalie Veber, et al. · Neuroendocrinology · 19
Blood–brain barrier and atrial natriuretic factor
1988 · P. E. Chabrier, P. Roubert, et al. · Canadian Journal of Physiology and Pharmacology · 18
Novel non-peptide ligands for the somatostatin sst3 receptor
2001 · Christophe Moinet, Marie-Odile Contour-Galcéra, et al. · Bioorganic & Medicinal Chemistry Letters · 17
Decrease in endothelin-1 renal receptors during the 1st month of life in the rat
1996 · Laurence Abadie, Isabelle Blazy, et al. · Pediatric Nephrology · 15
Upregulation of Renal Endothelin Receptors in Glycerol-Induced Acute Renal Failure in the Rat
1993 · P. Roubert, S. Cornet, et al. · Journal of Cardiovascular Pharmacology · 13
Binding Characteristics of Endothelin Isoforms (ET-1, ET-2, and ET-3) in Vascular Smooth Muscle Cells
1991 · P. Roubert, V. Gillard, et al. · Journal of Cardiovascular Pharmacology · 13
Receptor Regulation of Atrial Natriuretic Factor
2008 · P.E. Chabrier, P. Roubert, et al. · Blood Vessels · 10
Endothelin Receptors in Testosterone-Induced Prostatic Hypertrophy in Rats
1998 · Lydie Auger-Pourmarin, Pierre Roubert, et al. · The Japanese Journal of Pharmacology · 9
α1-Adrenoceptors in testosterone-induced prostatic hypertrophy
1998 · L Auger-Pourmarin, P Roubert, et al. · European Journal of Pharmacology · 8
Works count: 51
Citation count: 899
H-index: 18
I10-index: 23
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