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Author

Michael Edlund

Institution: Medivir (Sweden)
OpenAlex ID: A5110137214
In Vitro Resistance Profile of the Hepatitis C Virus NS3/4A Protease Inhibitor TMC435
2010 · Oliver Lenz, Thierry Verbinnen, et al. · Antimicrobial Agents and Chemotherapy · 218
In Vitro Activity and Preclinical Profile of TMC435350, a Potent Hepatitis C Virus Protease Inhibitor
2009 · Tse-I Lin, Oliver Lenz, et al. · Antimicrobial Agents and Chemotherapy · 195
Epidermal Overexpression of Stratum Corneum Chymotryptic Enzyme in Mice: A Model for Chronic Itchy Dermatitis
2002 · Assar Bäckman, Annelii Ny, et al. · Journal of Investigative Dermatology · 181
Structure–activity relationship study on a novel series of cyclopentane-containing macrocyclic inhibitors of the hepatitis C virus NS3/4A protease leading to the discovery of TMC435350
2008 · Pierre Raboisson, Herman de Kock, et al. · Bioorganic & Medicinal Chemistry Letters · 146
Induced‐Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target
2010 · Maxwell D. Cummings, Jimmy Lindberg, et al. · Angewandte Chemie International Edition · 98
Recombinant Human-Milk Bile-Salt-Stimulated Lipase. Functional Properties are Retained in the Absence of Glycosylation and the Unique Proline-Rich Repeats
1995 · Lars Blackberg, Mats Stromqvist, et al. · European Journal of Biochemistry · 37
BACE-1 inhibition prevents the γ-secretase inhibitor evoked Aβ rise in human neuroblastoma SH-SY5Y cells
2011 · Anne Jämsä, Oscar Belda, et al. · Journal of Biomedical Science · 27
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Synthesis and SAR of potent inhibitors of the Hepatitis C virus NS3/4A protease: Exploration of P2 quinazoline substituents
2010 · Magnus Nilsson, Anna Karin Belfrage, et al. · Bioorganic & Medicinal Chemistry Letters · 25
Discovery of novel, potent and bioavailable proline-urea based macrocyclic HCV NS3/4A protease inhibitors
2008 · Sandrine Vendeville, Magnus Nilsson, et al. · Bioorganic & Medicinal Chemistry Letters · 24
Recombinant human bile salt-stimulated lipase: an example of defectiveO-glycosylation of a protein produced in milk of transgenic mice
1996 · Mats Strömqvist, Jan Törnell, et al. · Transgenic Research · 23
Synthesis of potent BACE-1 inhibitors incorporating a hydroxyethylene isostere as central core
2009 · Fredrik Wångsell, Karin Gustafsson, et al. · European Journal of Medicinal Chemistry · 22
The resorptive apparatus of osteoclasts supports lysosomotropism and increases potency of basic versus non-basic inhibitors of cathepsin K
2010 · Karen Fuller, Erik Lindstrom, et al. · Bone · 13
Properties of recombinant human plasma procarboxypeptidase U produced in mammalian and insect cells
2004 · Mats Strömqvist, Lennart Hansson, et al. · Clinica Chimica Acta · 10
Inside Cover: Induced‐Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target (Angew. Chem. Int. Ed. 9/2010)
2010 · Maxwell D. Cummings, Jimmy Lindberg, et al. · Angewandte Chemie International Edition · 9
Induced‐Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target
2010 · Maxwell D. Cummings, Jimmy Lindberg, et al. · Angewandte Chemie · 5
Innentitelbild: Induced‐Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target (Angew. Chem. 9/2010)
2010 · Maxwell D. Cummings, Jimmy Lindberg, et al. · Angewandte Chemie · 1
Corrigendum: Induced‐Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target
2010 · Maxwell D. Cummings, Jimmy Lindberg, et al. · Angewandte Chemie International Edition
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Berichtigung: Induced‐Fit Binding of the Macrocyclic Noncovalent Inhibitor TMC435 to its HCV NS3/NS4A Protease Target
2010 · Maxwell D. Cummings, Jimmy Lindberg, et al. · Angewandte Chemie
Design and Synthesis of BACE-1 Inhibitors Containing a New Hydroxyethylene (HE) Scaffold: Potent activities in a cellular assay
2009 · Jenny Adrian Meredith, Catarina Björklund, et al.
Works count: 20
Citation count: 1,034
H-index: 12
I10-index: 13
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