Author

Seiji Tamura

Institution: Astellas Pharma (Japan)

Observed institution: Astellas Pharma (Japan)

OpenAlex ID: A5112082249

Radioligand Binding Properties and Pharmacological Characterization of 6-Amino-N-cyclohexyl-N,3-dimethylthiazolo[3,2-a]benzimidazole-2-carboxamide (YM-298198), a High-Affinity, Selective, and Noncompetitive Antagonist of Metabotropic Glutamate Receptor Type 1

2005 · Atsuyuki Kohara, Takashi Toya, et al. · Journal of Pharmacology and Experimental Therapeutics · 78

Neuroprotective effects of the selective type 1 metabotropic glutamate receptor antagonist YM-202074 in rat stroke models

2007 · Atsuyuki Kohara, Masayasu Takahashi, et al. · Brain Research · 68

Neurometer Measurement of Current Stimulus Threshold in Rats

2001 · Tetsuo Kiso, Yukinori Nagakura, et al. · Journal of Pharmacology and Experimental Therapeutics · 65

Minodronic acid, a third-generation bisphosphonate, antagonizes purinergic P2X2/3 receptor function and exerts an analgesic effect in pain models

2008 · Shuichiro Kakimoto, Yukinori Nagakura, et al. · European Journal of Pharmacology · 39

Antinociceptive profile of a selective metabotropic glutamate receptor 1 antagonist YM-230888 in chronic pain rodent models

2007 · Atsuyuki Kohara, Yukinori Nagakura, et al. · European Journal of Pharmacology · 22

AS1069562, the (+)-Isomer of Indeloxazine, Exerts Analgesic Effects in a Rat Model of Neuropathic Pain with Unique Characteristics in Spinal Monoamine Turnover

2013 · Nobuhito Murai, Toshiaki Aoki, et al. · Journal of Pharmacology and Experimental Therapeutics · 16

Antinociceptive effects of AS1069562, the (+)-isomer of indeloxazine, on spinal hypersensitivity induced by intrathecal injection of prostaglandin in mice: Comparison with duloxetine and amitriptyline

2014 · Nobuhito Murai, Mina Tsukamoto, et al. · European Journal of Pharmacology · 8

AS1069562, the (+)-isomer of indeloxazine, but not duloxetine has a curative-like analgesic effect in a rat model of streptozotocin-induced diabetic neuropathy

2013 · Nobuhito Murai, Toshiaki Aoki, et al. · Neuropharmacology · 8

Design, synthesis, and biological evaluation of novel biphenyl-4-carboxamide derivatives as orally available TRPV1 antagonists

2018 · Hiromasa Oka, Koichi Yonezawa, et al. · Bioorganic & Medicinal Chemistry · 6

AS1069562, the (+)-isomer of indeloxazine, exerts analgesic effects in rat models of nociceptive pain

2015 · Nobuhito Murai, Nobuaki Takeshita, et al. · Neurological Research · 1

Works count: 10

Citation count: 311

H-index: 8

I10-index: 6