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Enamine

Homepage URL: enamine.net
Alternate name: Enamine Ltd
Country: UA
ROR: 02t6zky14
Wikidata ID: entity/Q5375203
Crossref ID: 501100019003
DOI: 10.13039/501100019003
OpenAlex ID: F4320330169
Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses
2022 · Andreas Luttens, Hjalmar Gullberg, et al. · Journal of the American Chemical Society · 246
A Radical Approach to Anionic Chemistry: Synthesis of Ketones, Alcohols, and Amines
2019 · Shengyang Ni, Natalia M. Padial, et al. · Journal of the American Chemical Society · 228
Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2
2023 · Stefan Gahbauer, Galen J. Correy, et al. · Proceedings of the National Academy of Sciences · 133
Quaternary Centers by Nickel‐Catalyzed Cross‐Coupling of Tertiary Carboxylic Acids and (Hetero)Aryl Zinc Reagents
2019 · Tie‐Gen Chen, Haolin Zhang, et al. · Angewandte Chemie International Edition · 104
Rapid traversal of vast chemical space using machine learning-guided docking screens
2025 · Andreas Luttens, Israel Cabeza de Vaca, et al. · Nature Computational Science · 101
Electrochemical C(sp3)–H Fluorination
2019 · Yusuke Takahira, Miao Chen, et al. · Synlett · 100
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Late-Stage Saturation of Drug Molecules
2024 · De-Hai Liu, Philipp M. Pflüger, et al. · Journal of the American Chemical Society · 85
Saturated Boronic Acids, Boronates, and Trifluoroborates: An Update on Their Synthetic and Medicinal Chemistry
2021 · Dmitriy M. Volochnyuk, Alina O. Gorlova, et al. · Chemistry - A European Journal · 84
Design, synthesis and evaluation of novel sulfonamides as potential anticancer agents
2018 · Maryna V. Kachaeva, Diana M. Hodyna, et al. · Computational Biology and Chemistry · 75
γ-(S)-Trifluoromethyl proline: evaluation as a structural substitute of proline for solid state 19 F-NMR peptide studies
2015 · Vladimir Kubyshkin, Sergii Afonin, et al. · Organic & Biomolecular Chemistry · 68
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Three-component synthesis of fluorinated pyrazoles from fluoroalkylamines, NaNO 2 and electron-deficient alkynes
2015 · Pavel K. Mykhailiuk · Organic & Biomolecular Chemistry · 68
Synthesis of Spirocyclic Pyrrolidines: Advanced Building Blocks for Drug Discovery
2017 · Bohdan A. Chalyk, Maryna V. Butko, et al. · Chemistry - A European Journal · 64
Electron-Rich Amino Heterocyclesfor Regiospecific Synthesis of Trifluoromethyl-ContainingFused Pyridines
2003 · Dmitriy M. Volochnyuk, Alexei O. Pushechnikov, et al. · Synthesis · 59
Photooxygenation of an amino-thienopyridone yields a more potent PTP4A3 inhibitor
2016 · Joseph M. Salamoun, Kelley E. McQueeney, et al. · Organic & Biomolecular Chemistry · 54
Discovery and biological evaluation of adamantyl amide 11β-HSD1 inhibitors
2007 · Scott P. Webster, Peter Ward, et al. · Bioorganic & Medicinal Chemistry Letters · 53
Small molecule PGC-1α1 protein stabilizers induce adipocyte Ucp1 expression and uncoupled mitochondrial respiration
2018 · A.T. Pettersson-Klein, M. Izadi, et al. · Molecular Metabolism · 51
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Synthesis, anticancer and FGFR1 inhibitory activity of isoindolo[2,1-a][1,2,4]triazino[2,3-c]quinazoline derivatives
2016 · O. Yu. Voskoboynik, S. A. Starosyla, et al. · Medical and Clinical Chemistry · 50
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Impact of HDAC inhibitors on macrophage polarization to enhance innate immunity against infections
2024 · Mohammad Faizan Bhat, Sonja Srdanović, et al. · Drug Discovery Today · 49
Tackling recalcitrant Pseudomonas aeruginosa infections in critical illness via anti-virulence monotherapy
2022 · Vijay K. Singh, Marianna Almpani, et al. · Nature Communications · 48
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Synthesis of annulated benzimidazoles via amidine cyclization
2012 · Kostiantyn Liubchak, Kostiantyn Nazarenko, et al. · Tetrahedron · 48
Mapping the chemical chromatin reactivation landscape identifies BRD4-TAF1 cross-talk
2016 · Sara Sdelci, Charles-Hugues Lardeau, et al. · Nature Chemical Biology · 47
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Oxa-spirocycles: synthesis, properties and applications
2021 · Kateryna Fominova, Taras Diachuk, et al. · Chemical Science · 46
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Bicyclic Pyrrolidines for Medicinal Chemistry via [3 + 2]-Cycloaddition
2021 · Vladimir I. Savych, Vladimir L. Mykhalchuk, et al. · The Journal of Organic Chemistry · 45
Three-component synthesis of C2F5-substituted pyrazoles from C2F5CH2NH2·HCl, NaNO2 and electron-deficient alkynes
2015 · Pavel K Mykhailiuk · Beilstein Journal of Organic Chemistry · 45
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Radical Reactions of Alkyl 2‑Bromo-2,2-difluoroacetates with Vinyl Ethers: “Omitted” Examples and Application for the Synthesis of 3,3-Difluoro-GABA
2015 · Ivan S. Kondratov, Maksym Ya. Bugera, et al. · The Journal of Organic Chemistry · 44
Works count: 401
Citation count: 4,935
H-index: 34
I10-index: 137
2-year mean citedness: 4.01
Awards count: 0
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