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Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2-d]pyrimidines as EGFR and ErbB-2 inhibitors

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Year: 2008
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2008.11.023
Authors: Kirk L. Stevens, Krystal J. Alligood, Jennifer G. Badiang Alberti, Thomas R. Caferro, Stanley D. Chamberlain, Scott H. Dickerson, Hamilton D. Dickson, Holly K. Emerson, Robert J. Griffin, Robert D. Hubbard, Barry R. Keith, Robert J. Mullin, Kimberly G. Petrov, Roseanne M. Gerding, Michael J. Reno, Tara R. Rheault, David W. Rusnak, Douglas M. Sammond, Stephon C. Smith, David E. Uehling, Alex G. Waterson, Edgar R. Wood
Institution: GlaxoSmithKline (United States)
Language: English

Topic: Synthesis and biological activity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: green
OpenAlex ID: W1972920012
FWCI: 0.495
Cites: 17
Cited by: 21
Related to: 10
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