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Discovery of an Opioid κ Receptor Selective Pure Antagonist from a Library of N-Substituted 4β-Methyl-5-(3-hydroxyphenyl)morphans

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Year: 2002
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm020084h
Authors: James B. Thomas, Robert N. Atkinson, Nivedita Namdev, Richard B. Rothman, Kenneth M. Gigstad, Scott E. Fix, S. Wayne Mascarella, Jason P. Burgess, N. Ariane Vinson, Heng Xu, Christina M. Dersch, Buddy E. Cantrell, Dennis M. Zimmerman, F. Ivy Carroll
Institutions: National Institute on Drug Abuse, Eli Lilly (United States), RTI International
Language: English

Topic: Neuropeptides and Animal Physiology
Subfield: Cellular and Molecular Neuroscience
Field: Neuroscience
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: National Institute on Drug Abuse
Awards: G3861717303, Selective Opioid Antagonists as Medications for Drug Abuse
OpenAlex ID: W1996795014
FWCI: 1.278
Cites: 10
Cited by: 29
Related to: 10
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