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Structure–activity relationships of a novel pyranopyridine series of Gram-negative bacterial efflux pump inhibitors

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Year: 2015
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2015.03.016
Authors: Son T. Nguyen, Steven M. Kwasny, Xiaoyuan Ding, Steven C. Cardinale, Courtney T. McCarthy, Hong-Suk Kim, Hiroshi Nikaido, Norton P. Peet, John D. Williams, Terry L. Bowlin, Timothy J. Opperman
Institutions: Microbiotix (United States), University of California, Berkeley
Language: English

Topic: Antibiotic Resistance in Bacteria
Subfield: Molecular Medicine
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: green

Funder: National Institute of Allergy and Infectious Diseases
Awards: Optimization of novel pyranopyridine efflux pump inhibitors, Optimization of novel pyranopyridine efflux pump inhibitors
OpenAlex ID: W2015050900
FWCI: 4.418
Cites: 41
Cited by: 84
Related to: 10
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