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Sulforaphane is not an effective antagonist of the human pregnane X-receptor in vivo

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Year: 2012
Type: article
Study design: Clinical Trial
Source: Toxicology and Applied Pharmacology
DOI: 10.1016/j.taap.2012.10.029
Authors: Emma Jane Poulton, Lisa Levy, Johanna W. Lampe, Danny D. Shen, Julia Tracy, Margaret C. Shuhart, Kenneth E. Thummel, David L. Eaton
Institutions: University of Washington, Fred Hutch Cancer Center
Language: English

Topic: Pharmacogenetics and Drug Metabolism
Subfield: Pharmacology
Field: Pharmacology, Toxicology and Pharmaceutics
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: green

Funders: Johns Hopkins University, Georgia Clinical and Translational Science Alliance, National Institutes of Health, U.S. Public Health Service, National Cancer Institute, National Institute of General Medical Sciences, National Institute of Environmental Health Sciences, National Center for Research Resources
Awards: Drug Interactions, Institute for Translational Health Science (UL1), Isothiocyanates as specific antagonists of human SXR, G5698425088, G5887241755, Hormonal Regulation of Human CYP3A, G71829041, Environmental Pathology/Toxicology Training Program, University of Washington Interdisciplinary Center for Exposures, Diseases, Genomics & Environment, Interdisciplinary Training in Cancer Research
OpenAlex ID: W2019810831
FWCI: 2.397
Cites: 51
Cited by: 40
Related to: 10
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