Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model▽
Year: 2008
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm800310g
Authors: Lisa D. Julian, Zhulun Wang, Tracy Bostick, Seb Caille, Rebekah Choi, Michael DeGraffenreid, Yongmei Di, Xiao He, Randall W. Hungate, Juan C. Jaen, Jinsong Liu, Mario Monshouwer, Dustin McMinn, Yosup Rew, Athena Sudom, Daqing Sun, Hua Tu, Stefania Ursu, Nigel Walker, Xuelei Yan, Qiuping Ye, Jay P. Powers
Institution: Amgen (United States)
Language: English
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
Open Access status: closed
OpenAlex ID: W2029301873
