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Design, synthesis, and biological evaluation of novel histone deacetylase 1 inhibitors through click chemistry

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Year: 2013
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2013.03.102
Authors: Qiao Sun, Yiwu Yao, Chunping Liu, Hua Li, Hequan Yao, Xiaowen Xue, Jinsong Liu, Zhengchao Tu, Sheng Jiang
Institutions: Chinese Academy of Sciences, Guangzhou Institutes of Biomedicine and Health, China Pharmaceutical University
Language: English

Topic: Histone Deacetylase Inhibitors Research
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Science Foundation, National Natural Science Foundation of China, National Key Research and Development Program of China
Awards: Argyrin A 的全合成研究, G2922681079, 组蛋白去乙酰化酶抑制剂Lar-7的构效关系及其抗肿瘤活性的研究
OpenAlex ID: W2060054861
FWCI: 1.046
Cites: 29
Cited by: 18
Related to: 10
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