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Proteasome Regulator Marizomib (NPI-0052) Exhibits Prolonged Inhibition, Attenuated Efflux, and Greater Cytotoxicity than Its Reversible Analogs

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Year: 2011
Type: article
Source: Journal of Pharmacology and Experimental Therapeutics
DOI: 10.1124/jpet.110.177824
Authors: Amanda Obaidat, Jeffrey Weiss, Brett Wahlgren, Rama R. Manam, Venkat R. Macherla, Katherine McArthur, Ta-Hsiang Chao, Michael A. Palladino, G. Kenneth Lloyd, Barbara C. Potts, Salvatore J. Enna, Saskia T.C. Neuteboom, Bruno Hagenbuch
Institutions: University of Kansas Medical Center, The University of Kansas Cancer Center
Language: English

Topic: Ubiquitin and proteasome pathways
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: American Association for Cancer Research, National Institutes of Health, National Institute of General Medical Sciences, National Institute of Environmental Health Sciences, National Center for Research Resources
Awards: G1958400685, G2850908965, Nuclear Receptors in Liver Health and Disease, G4686375030, Molecular Characterization of Hepatic Organic Anion Transporting Polypeptides, Training Program in Environmental Toxicology, G9000099149
OpenAlex ID: W2072898309
FWCI: 2.193
Cites: 22
Cited by: 32
Related to: 10
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