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Design, Synthesis, and Evaluation of Aza-Peptide Michael Acceptors as Selective and Potent Inhibitors of Caspases-2, -3, -6, -7, -8, -9, and -10

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Year: 2006
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm0601405
Authors: Özlem Doǧan Ekici, Zhao Zhao Li, Amy J. Campbell, Karen Ellis James, Juliana L. Asgian, Jowita Mikolajczyk, Guy S. Salvesen, Rajkumar Ganesan, Stjepan Jelakovic, Markus G. Grütter, James C. Powers
Institutions: Georgia Institute of Technology, Sanford Burnham Prebys Medical Discovery Institute, University of Zurich
Language: English

Topic: Cell death mechanisms and regulation
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: closed

Funder: National Institute of General Medical Sciences
Award: CASPASE INHIBITORS
OpenAlex ID: W2087578110
FWCI: 1.684
Cites: 34
Cited by: 78
Related to: 10
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