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Synthesis and optimization of thiadiazole derivatives as a novel class of substrate competitive c-Jun N-terminal kinase inhibitors

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Year: 2009
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2009.12.013
Authors: Surya K. De, Vida Chen, John L. Stebbins, Li-Hsing Chen, Jason F. Cellitti, Thomas Machleidt, Elisa Barile, Megan Riel-Mehan, Russell Dahl, Li Yang, Aras Emdadi, Ria Murphy, Maurizio Pellecchia
Institution: Sanford Burnham Prebys Medical Discovery Institute
Language: English

Topic: Synthesis and biological activity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences

Open Access status: green

Funders: National Institutes of Health, National Institute of Diabetes and Digestive and Kidney Diseases
Awards: G5394619753, G5734286822, G7399545639, Allosteric JNK modulators for the treatment of diabetes
OpenAlex ID: W2087774017
FWCI: 1.934
Cites: 28
Cited by: 25
Related to: 10
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