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Oxindole-Based Inhibitors of Cyclin-Dependent Kinase 2 (CDK2): Design, Synthesis, Enzymatic Activities, and X-ray Crystallographic Analysis

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Year: 2001
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm010117d
Authors: H. Neal Bramson, John Corona, Stephen T. Davis, Scott H. Dickerson, Mark Edelstein, Stephen V. Frye, Robert T. Gampe, Phil A. Harris, Anne Hassell, William D. Holmes, Robert N. Hunter, Karen E. Lackey, Brett Lovejoy, Michael J. Luzzio, Val Montana, Warren J. Rocque, David Rusnak, Lisa Shewchuk, James M. Veal, Duncan H. Walker, Lee F. Kuyper
Institution: GlaxoSmithKline (United States)
Language: English

Topic: Heterocyclic Compound Synthesis and Bioactivity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2117263757
FWCI: 9.789
Cites: 41
Cited by: 277
Related to: 10
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