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Cellular Inhibition of Checkpoint Kinase 2 (Chk2) and Potentiation of Camptothecins and Radiation by the Novel Chk2 Inhibitor PV1019 [7-Nitro-1H-indole-2-carboxylic acid {4-[1-(guanidinohydrazone)-ethyl]-phenyl}-amide]

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Year: 2009
Type: article
Source: Journal of Pharmacology and Experimental Therapeutics
DOI: 10.1124/jpet.109.154997
Authors: Andrew G. Jobson, George T. Lountos, Philip L. Lorenzi, Jenny Llamas, John Connelly, David Cerna, Joseph E. Tropea, Akikazu Onda, Gabriele Zoppoli, Sudhir Kondapaka, Guangtao Zhang, Natasha J. Caplen, John H. Cardellina, Stephen S. Yoo, Anne Monks, Christopher Self, David S. Waugh, Robert H. Shoemaker, Yves Pommier
Institutions: National Institutes of Health, National Cancer Institute, Center for Cancer Research, Provid Pharmaceuticals (United States), National Cancer Institute, National Cancer Institute
Language: English

Topic: DNA Repair Mechanisms
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: U.S. Department of Energy, National Institutes of Health, Office of Science, National Heart, Lung, and Blood Institute, National Cancer Institute, Basic Energy Sciences, Argonne National Laboratory
OpenAlex ID: W2117389132
FWCI: 2.285
Cites: 41
Cited by: 95
Related to: 10
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