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Oxime esters as selective, covalent inhibitors of the serine hydrolase retinoblastoma-binding protein 9 (RBBP9)

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Year: 2010
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2010.02.011
Authors: Daniel A. Bachovchin, Monique R. Wolfe, Kim Masuda, Steven J. Brown, Timothy P. Spicer, Virneliz Fernandez-Vega, Peter Chase, Peter S. Hodder, Hugh Rosen, Benjamin F. Cravatt
Institution: Scripps Research Institute
Language: English

Topic: Protease and Inhibitor Mechanisms
Subfield: Cancer Research
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: green

Funders: National Institute of Mental Health, National Cancer Institute
Awards: The Comprehensive Center for Chemical Probe Discovery and Optimization at Scripps, G3510558551, G6296143508, G6838120957
OpenAlex ID: W2130829883
FWCI: 1.083
Cites: 22
Cited by: 30
Related to: 10
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