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Preferred Binding Orientations of Phenacetin in CYP1A1 and CYP1A2 Are Associated with Isoform-Selective Metabolism

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Year: 2012
Type: article
Source: Drug Metabolism and Disposition
DOI: 10.1124/dmd.112.047308
Authors: Qingbiao Huang, Rahul S. Deshmukh, Spencer S. Ericksen, Youbin Tu, Grazyna D. Szklarz
Institution: West Virginia University
Language: English

Topic: Pharmacogenetics and Drug Metabolism
Subfield: Pharmacology
Field: Pharmacology, Toxicology and Pharmaceutics
Domain: Life Sciences

Open Access status: bronze

Funders: West Virginia University, National Institutes of Health, National Institute of General Medical Sciences, National Center for Research Resources
Awards: G2345570189, G449543902, Cobre for Signal Transduction and Cancer, G580369581, Cytochrome P450-reductase interactions in P450 1A subfamily, G9000062380
OpenAlex ID: W2140647339
FWCI: 1.445
Cites: 41
Cited by: 24
Related to: 10
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