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A Single Glycine in Extracellular Loop 1 Is the Critical Determinant for Pharmacological Specificity of Dopamine D2 and D3 Receptors

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Year: 2013
Type: article
Source: Molecular Pharmacology
DOI: 10.1124/mol.113.087833
Authors: Mayako Michino, Prashant Donthamsetti, Thijs Beuming, Ashwini Banala, Lihua Duan, Thomas Roux, Yang Han, Eric Trinquet, Amy Hauck Newman, Jonathan A. Javitch, Lei Shi
Institutions: National Institutes of Health, National Institute on Drug Abuse, Schrodinger (United States), Cornell University, Columbia University Irving Medical Center, Cisbio (France), Weill Cornell Medicine, New York State Psychiatric Institute, Columbia University
Language: English

Topic: Receptor Mechanisms and Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: bronze

Funders: National Institutes of Health, National Institute of Mental Health, National Institute on Drug Abuse
Awards: Molecular determinants for the action of psychostimulants, The Neurotransmitter: Sodium Symporter Permeation Pathway, G521840061, G9000068177, G9000283290, G900070601, Structure and Function of Dopamine Receptors, G94731328
OpenAlex ID: W2151088690
FWCI: 3.092
Cites: 47
Cited by: 72
Related to: 10
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