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Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38

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Year: 2015
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.5b00992
Authors: J. David Becherer, Eric E. Boros, Tiffany Y. Carpenter, David J. Cowan, David N. Deaton, Curt D. Haffner, Michael R. Jeune, Istvan W. Kaldor, J. Chuck Poole, Frank Preugschat, Tara R. Rheault, Christie A. Schulte, Barry G. Shearer, Todd W. Shearer, Lisa M. Shewchuk, Terrence L. Smalley, Eugene L. Stewart, J. Darren Stuart, John C. Ulrich
Institution: GlaxoSmithKline (United States)
Language: English

Topic: Sirtuins and Resveratrol in Medicine
Subfield: Geriatrics and Gerontology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2225399376
FWCI: 3.732
Cites: 23
Cited by: 54
Related to: 10
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