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8-Tetrahydropyran-2-yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors

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Year: 2014
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/jm5015132
Authors: Allen A. Thomas, Kevin W. Hunt, Brad Newhouse, Ryan J. Watts, Xingrong Liu, Guy Vigers, Darin Smith, Susan P. Rhodes, Karin D. Brown, Jennifer N. Otten, Michael Burkard, April A. Cox, Mary K. Geck Do, Darrin Dutcher, Sumeet Rana, Robert K. DeLisle, Kelly Regal, Albion D. Wright, Robert Groneberg, Jiangpeng Liao, Kimberly Scearce-Levie, Michael Siu, Hans E. Purkey, Joseph P. Lyssikatos
Institutions: Array BioPharma (United States), Genentech, WuXi AppTec (China)
Language: English

Topic: Alzheimer's disease research and treatments
Subfield: Physiology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2334222265
FWCI: 2.216
Cites: 50
Cited by: 19
Related to: 10
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