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Discovery and development of benzo-[1,2,4]-triazolo-[1,4]-oxazepine GPR142 agonists for the treatment of diabetes

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Year: 2016
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2016.04.018
Authors: Jonathan E. Wilson, Ravi Kurukulasuriya, Christopher Sinz, Matthew Lombardo, Kate Bender, Dann Parker, Edward C. Sherer, Melissa Costa, Karen Dingley, Xiaofang Li, Stanley Mitelman, Sharon Tong, Randal Bugianesi, Anka Ehrhardt, Birgit Priest, Kevin Ratliff, Feroze Ujjainwalla, Ravi Nargund, William K. Hagmann, Scott Edmondson
Institution: Merck & Co., Inc., Rahway, NJ, USA (United States)
Language: English

Topic: Diabetes Treatment and Management
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2405189531
FWCI: 3.013
Cites: 21
Cited by: 18
Related to: 10
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