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Optimization of pyrazole-containing 1,2,4-triazolo-[3,4-b]thiadiazines, a new class of STAT3 pathway inhibitors

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Year: 2016
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2016.06.017
Authors: Matthew G. LaPorte, Zhuzhu Wang, Raffaele Colombo, Atefeh Garzan, Vsevolod A. Peshkov, Mary Liang, Paul A. Johnston, Mark E. Schurdak, Malabika Sen, Daniel P. Camarco, Yun Hua, Netanya I. Pollock, John S. Lazo, Jennifer R. Grandis, Peter Wipf, Donna M. Huryn
Institutions: University of Pittsburgh, UPMC Hillman Cancer Center, University of Virginia, University of California, San Francisco
Language: English

Topic: Cytokine Signaling Pathways and Interactions
Subfield: Oncology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: green

Funder: National Cancer Institute
Awards: G34221693, G386607036
OpenAlex ID: W2411377232
FWCI: 1.86
Cites: 27
Cited by: 31
Related to: 10
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