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Evaluation of 7-arylaminopyrazolo[1,5-a]pyrimidines as anti-Plasmodium falciparum, antimalarial, and Pf-dihydroorotate dehydrogenase inhibitors

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Year: 2016
Type: article
Source: European Journal of Medicinal Chemistry
DOI: 10.1016/j.ejmech.2016.09.073
Authors: Luís Felipe S.P. Azeredo, Julia P. Coutinho, Valquiria A.P. Jabor, Patricia R. Feliciano, Maria Cristina Nonato, Carlos R. Kaiser, Carla Maria S. Menezes, Amanda S.O. Hammes, Ernesto Raul Caffarena, Lucas V.B. Hoelz, Nicolli B. de Souza, Glaécia A.N. Pereira, Isabela P. Cerávolo, Antoniana U. Krettli, Nubia Boechat
Institutions: Universidade Federal do Rio de Janeiro, Instituto de Tecnologia em Fármacos, Fundação Oswaldo Cruz, Universidade Federal de Minas Gerais, Fiocruz Minas, Universidade de São Paulo
Language: English

Topic: Malaria Research and Control
Subfield: Public Health, Environmental and Occupational Health
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Fundação de Amparo à Pesquisa do Estado de São Paulo, Coordenação de Aperfeiçoamento de Pessoal de Nível Superior
Award: Development of leishmanicidal drugs based on the selective inhibition of the enzyme dihydroorotate dehydrogenase
OpenAlex ID: W2529330909
FWCI: 7.604
Cites: 38
Cited by: 84
Related to: 10
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