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Discovery of orally active hepatoselective glucokinase activators for treatment of Type II Diabetes Mellitus

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Year: 2016
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2016.10.088
Authors: Jiayi Xu, Songnian Lin, Robert W. Myers, Maria E. Trujillo, Michele J. Pachanski, Sunita Malkani, Hsuan-shen Chen, Zhesheng Chen, Brian Campbell, George J. Eiermann, Nadine Elowe, Brian T. Farrer, Wen Feng, Qinghong Fu, Roman Kats-Kagan, Michael Kavana, Daniel R. McMasters, Kaushik Mitra, Xinchun Tong, Libo Xu, Fengqi Zhang, Rui Zhang, George H. Addona, Joel P. Berger, Bei Zhang, Emma R. Parmee
Institution: Merck & Co., Inc., Rahway, NJ, USA (United States)
Language: English

Topic: Diabetes Treatment and Management
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2544680916
FWCI: 1.673
Cites: 43
Cited by: 13
Related to: 10
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