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Functions of bromodomain-containing proteins and their roles in homeostasis and cancer

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Year: 2017
Type: review
Source: Nature Reviews Molecular Cell Biology
DOI: 10.1038/nrm.2016.143
Authors: Takao Fujisawa, Panagis Filippakopoulos
Institution: Ludwig Cancer Research
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: green

Funders: Pfizer, Genome Canada, Ludwig Institute for Cancer Research, Wellcome Trust, European Federation of Pharmaceutical Industries and Associations, Ontario Ministry of Economic Development and Innovation, Fundação de Amparo à Pesquisa do Estado de São Paulo, Innovative Medicines Initiative, Novartis Pharma, Medical Research Council
Awards: Open access research to promote drug discovery., A UK Hub to Catalyse Open Target Discovery., G3603401286, ZMYND8-regulation of MITF as potential therapeutic target in melanoma, G7669079602, Structural role of BET bromodomains in transcription.
OpenAlex ID: W2568322231
FWCI: 5.081
Cites: 188
Cited by: 612
Related to: 10
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