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Ligand and Target Discovery by Fragment-Based Screening in Human Cells

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Year: 2017
Type: article
Source: Cell
DOI: 10.1016/j.cell.2016.12.029
Authors: Christopher G. Parker, Andrea Galmozzi, Yujia Wang, Bruno E. Correia, Kenji Sasaki, Christopher M. Joslyn, Arthur S. Kim, Cullen L. Cavallaro, R. Michael Lawrence, Stephen R. Johnson, Iñigo Narvaiza, Enrique Saez, Benjamin F. Cravatt
Institutions: Scripps Research Institute, École Polytechnique Fédérale de Lausanne, Bristol-Myers Squibb (United States), Salk Institute for Biological Studies
Language: English

Topic: Click Chemistry and Applications
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: American Cancer Society, American Heart Association, National Institutes of Health, National Cancer Institute, National Institute of Diabetes and Digestive and Kidney Diseases
Awards: G3510558551, Seahorse XF96 Extracellular Flux Analyzer, Identification and Therapeutic Valiation of Adipocyte Serine Hydrolases of Metab, G6799995778, G921902380
OpenAlex ID: W2575838842
FWCI: 18.68
Cites: 59
Cited by: 434
Related to: 10
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