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A Phase 1 Study of the DOT1L Inhibitor, Pinometostat (EPZ-5676), in Adults with Relapsed or Refractory Leukemia: Safety, Clinical Activity, Exposure and Target Inhibition

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Year: 2015
Type: article
Study design: Clinical Trial
Source: Blood
DOI: 10.1182/blood.v126.23.2547.2547
Authors: Eytan M. Stein, Guillermo Garcia-Manero, David A. Rizzieri, Raoul Tibes, Jesus G. Berdeja, Mojca Jongen-Lavrencic, Jessica K. Altman, Hartmut Dohner, Blythe Thomson, Stephen J. Blakemore, Scott Daigle, Greg Fine, Nigel J. Waters, Andrei V Krivstov, Richard Koche, Scott A. Armstrong, Peter T Ho, Bob Lowenberg, Martin S Tallman
Institutions: Memorial Sloan Kettering Cancer Center, The University of Texas MD Anderson Cancer Center, Duke Medical Center, Mayo Clinic in Arizona, Sarah Cannon, Erasmus MC, Northwestern University, University Hospital Ulm, Epizyme (United States)
Language: English

Topic: Acute Myeloid Leukemia Research
Subfield: Hematology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2584347108
FWCI: 5.88
Cites:
Cited by: 47
Related to: 10
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