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Structural Biology-Inspired Discovery of Novel KRAS–PDEδ Inhibitors

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Year: 2017
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.7b01243
Authors: Yan Jiang, Chunlin Zhuang, Long Chen, Junjie Lu, Guoqiang Dong, Zhenyuan Miao, Wannian Zhang, Jian Li, Chunquan Sheng
Institutions: Second Military Medical University, East China University of Science and Technology
Language: English

Topic: Phosphodiesterase function and regulation
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: closed

Funders: Natural Science Foundation of Shanghai, National Natural Science Foundation of China, Shanghai Education Development Foundation, Shanghai Municipal Education Commission, Shanghai Municipal Health and Family Planning Commission
Awards: 蛋白-蛋白相互作用小分子探针设计、合成和生物活性研究, G1802630984, G3197000548, G5315190886
OpenAlex ID: W2755409777
FWCI: 0.992
Cites: 28
Cited by: 34
Related to: 10
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