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Identification of lead compounds for inhibitor design against tyrosyl DNA phosphodiesterase I by crystallographic fragment screening

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Year: 2017
Type: article
Source: Acta Crystallographica Section A Foundations and Advances
DOI: 10.1107/s0108767317097938
Authors: George T. Lountos, Xue Zhi Zhao, Evgeny Kiselev, Joseph E. Tropea, Danielle Needle, Terrence R. Burke, Yves Pommier, David S. Waugh
Institutions: Frederick National Laboratory for Cancer Research, National Cancer Institute, Leidos Biomedical Research Inc. (United States), National Cancer Institute, National Cancer Institute
Language: English

Topic: Enzyme Structure and Function
Subfield: Materials Chemistry
Field: Materials Science
Domain: Physical Sciences

Open Access status: bronze
OpenAlex ID: W2776594387
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Related to: 10
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