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Umbralisib, a novel PI3Kδ and casein kinase-1ε inhibitor, in relapsed or refractory chronic lymphocytic leukaemia and lymphoma: an open-label, phase 1, dose-escalation, first-in-human study

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Year: 2018
Type: article
Study design: Clinical Trial
Source: The Lancet Oncology
DOI: 10.1016/s1470-2045(18)30082-2
Authors: Howard A Burris, Ian W Flinn, Manish R Patel, Timothy S Fenske, Changchun Deng, Danielle M Brander, Martin Gutierrez, James H Essell, John G Kuhn, Hari P Miskin, Peter Sportelli, Michael S Weiss, Swaroop Vakkalanka, Michael R Savona, Owen A O'Connor
Institutions: Sarah Cannon, Tennessee Oncology, Medical College of Wisconsin, NewYork–Presbyterian Hospital, Columbia University Irving Medical Center, Columbia University, Duke Medical Center, Hackensack University Medical Center, Oncology Hematology Care, The University of Texas at San Antonio Health Science Center, TG Therapeutics, Inc. (United States), Rhizen Pharmaceuticals (Switzerland), Vanderbilt University Medical Center
Language: English

Topic: Chronic Lymphocytic Leukemia Research
Subfield: Genetics
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Bristol-Myers Squibb, TG Therapeutics
OpenAlex ID: W2788838674
FWCI: 17.54
Cites: 31
Cited by: 209
Related to: 10
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