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Chiral analogues of (+)-cyclazosin as potent α1B-adrenoceptor selective antagonist

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Year: 2018
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2018.05.023
Authors: Gianni Sagratini, Michela Buccioni, Gabriella Marucci, Elena Poggesi, Matthew Skorski, Stefano Costanzi, Dario Giardinà
Institutions: Università di Camerino, Recordati (Italy), American University
Language: English

Topic: Receptor Mechanisms and Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: bronze

Funders: National Science Foundation, Università degli Studi di Camerino, National Institute of General Medical Sciences
Awards: MRI: Acquisition of HPC at AU (Expanding Capabilities for Research and Research Training at American University through Shared High-Performance Computing), Enabling the application of Virtual Screening to GPCR Homology Models
OpenAlex ID: W2803607030
FWCI: 0.267
Cites: 39
Cited by: 5
Related to: 10
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