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Modulating PCAF/GCN5 Immune Cell Function through a PROTAC Approach

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Year: 2018
Type: article
Source: ACS Chemical Biology
DOI: 10.1021/acschembio.8b00705
Authors: Zuni I. Bassi, Martin C. Fillmore, Afjal H. Miah, Trevor D. Chapman, Claire Maller, Emma J. Roberts, Lauren C. Davis, Darcy E. Lewis, Nicholas W. Galwey, Kirsty E. Waddington, Valentino Parravicini, Abigail L. Macmillan-Jones, Celine Gongora, Philip G. Humphreys, Ian Churcher, Rab K. Prinjha, David F. Tough
Institutions: GlaxoSmithKline (United Kingdom), Inserm, Université de Montpellier, Institut de Recherche en Cancérologie de Montpellier
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2891213440
FWCI: 6.585
Cites: 21
Cited by: 185
Related to: 10
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