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Potent HIV-1 protease inhibitors incorporating squaramide-derived P2 ligands: Design, synthesis, and biological evaluation

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Year: 2019
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2019.08.006
Authors: Arun K. Ghosh, Jacqueline N. Williams, Satish Kovela, Jun Takayama, Hannah M. Simpson, D. Eric Walters, Shin-ichiro Hattori, Manabu Aoki, Hiroaki Mitsuya
Institutions: Purdue University West Lafayette, Rosalind Franklin University of Medicine and Science, National Center for Global Health and Medicine, National Institutes of Health, National Cancer Institute, Kumamoto University Hospital
Language: English

Topic: HIV/AIDS drug development and treatment
Subfield: Infectious Diseases
Field: Medicine
Domain: Health Sciences

Open Access status: green

Funders: Purdue University Center for Cancer Research, National Institutes of Health, National Institute of General Medical Sciences, National Institute of Allergy and Infectious Diseases
Awards: DESIGN AND SYNTHESIS OF NONPEPTIDE PROTEASE INHIBITORS, Design & Synthesis of Nonpeptide Protease Inhibitors, Design & Synthesis of Nonpeptide Protease Inhibitors, G9000252667
OpenAlex ID: W2965106829
FWCI: 1.533
Cites: 37
Cited by: 11
Related to: 10
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