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Recent Advances in Selective and Irreversible Covalent Ligand Development and Validation

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Year: 2019
Type: review
Source: Cell chemical biology
DOI: 10.1016/j.chembiol.2019.09.012
Authors: Tinghu Zhang, John M. Hatcher, Mingxing Teng, Nathanael S. Gray, Milka Kostic
Institutions: Harvard University, Dana-Farber Cancer Institute, Dana-Farber/Harvard Cancer Center
Language: English

Topic: Click Chemistry and Applications
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: Astellas Pharma US, Novartis, Sanofi, Taiho Pharmaceutical, National Institutes of Health, National Cancer Institute, Janssen Pharmaceuticals
Award: Targeting ALK through Degradation and Allosteric Inhibitors
OpenAlex ID: W2980410567
FWCI: 1.61
Cites: 88
Cited by: 178
Related to: 10
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