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First-generation structure-activity relationship studies of 2,3,4,9-tetrahydro-1H-carbazol-1-amines as CpxA phosphatase inhibitors

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Year: 2019
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2019.05.003
Authors: Yangxiong Li, Jessi J. Gardner, Katherine R. Fortney, Inga V. Leus, Vincent Bonifay, Helen I. Zgurskaya, Alexandre A. Pletnev, Sheng Zhang, Zhong-Yin Zhang, Gordon W. Gribble, Stanley M. Spinola, Adam S. Duerfeldt
Institutions: University of Oklahoma, Indiana University Indianapolis, Indiana University School of Medicine, Dartmouth College, Purdue University West Lafayette, Indiana University – Purdue University Indianapolis
Language: English

Topic: Bacterial Genetics and Biotechnology
Subfield: Genetics
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences

Open Access status: green

Funders: National Institutes of Health, National Cancer Institute, National Institute of Allergy and Infectious Diseases, National Center for Research Resources, National Center for Advancing Translational Sciences
Awards: Indiana Clinical and Translational Sciences Institute, Development of SHP2 inhibitors for targeted anti-cancer therapy, Predictive Models for Small-Molecule Accumulation in Gram-Negative Bacteria
OpenAlex ID: W2944694761
FWCI: 1.656
Cites: 23
Cited by: 15
Related to: 10
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