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Antibody-mediated delivery of chimeric protein degraders which target estrogen receptor alpha (ERα)

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Year: 2019
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2019.126907
Authors: Peter S. Dragovich, Pragya Adhikari, Robert A. Blake, Nicole Blaquiere, Jinhua Chen, Yun-Xing Cheng, Willem den Besten, Jinping Han, Steven J. Hartman, Jintang He, Mingtao He, Ellen Rei Ingalla, Amrita V. Kamath, Tracy Kleinheinz, Tommy Lai, Douglas D. Leipold, Chun Sing Li, Qi Liu, Jiawei Lu, Ying Lu, Fanwei Meng, Lingyao Meng, Carl Ng, Kaishan Peng, Gail Lewis Phillips, Thomas H. Pillow, Rebecca K. Rowntree, Jack D. Sadowsky, Deepak Sampath, Leanna Staben, Steven T. Staben, John Wai, Kunpeng Wan, Xinxin Wang, BinQing Wei, Ingrid E. Wertz, Jianfeng Xin, Keyang Xu, Hui Yao, Richard Zang, Donglu Zhang, Hao Zhou, Yongxin Zhao
Institutions: Genentech, WuXi AppTec (China), Pharmaron (China)
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W2994869094
FWCI: 3.123
Cites: 54
Cited by: 120
Related to: 10
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