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Advances in therapeutic peptides targeting G protein-coupled receptors

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Year: 2020
Type: review
Source: Nature Reviews Drug Discovery
DOI: 10.1038/s41573-020-0062-z
Authors: Anthony P. Davenport, Conor C. G. Scully, Chris de Graaf, Alastair J. H. Brown, Janet J. Maguire
Institutions: University of Cambridge, Addenbrooke's Hospital
Language: English

Topic: Receptor Mechanisms and Signaling
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: Wellcome Trust, Medical Research Council, NIHR Cambridge Biomedical Research Centre
Awards: Identification of 'hit to lead' small molecule biased' apelin receptor agonists for treating pulmonary arterial hypertension (PAH) using HTS and molecular modelling., G4576965740, Cambridge Confidence in Concepts: translating pathophysiological insights for patient benefit, G6868616705
OpenAlex ID: W3001942526
FWCI: 3.882
Cites: 209
Cited by: 283
Related to: 10
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