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Discovery of cyclic guanidine-linked sulfonamides as inhibitors of LMTK3 kinase

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Year: 2020
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2020.127108
Authors: Maria A. Ortiz, Heather Michaels, Brandon Molina, Sean Toenjes, Jennifer Davis, Guya Diletta Marconi, David Hecht, Jeffrey L. Gustafson, F. Javier Piedrafita, Adel Nefzi
Institutions: San Diego State University, Torrey Pines Institute For Molecular Studies, University of Chieti-Pescara, Southwestern College - California, Florida International University
Language: English

Topic: Computational Drug Discovery Methods
Subfield: Computational Theory and Mathematics
Field: Computer Science
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Institute for Health and Care Research, National Institutes of Health, National Cancer Institute
Awards: G4144886700, LMTK3 inhibitors for the treatment of breast cancer, G7471451890
OpenAlex ID: W3011673336
FWCI: 0.745
Cites: 35
Cited by: 12
Related to: 10
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