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Synthesis and structure–activity relationship studies of LLY-507 analogues as SMYD2 inhibitors

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Year: 2020
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
Authors: Bin Zhang, Liping Liao, Fan Wu, Fengcai Zhang, Zhongya Sun, Haijun Chen, Cheng Luo
Institutions: Fuzhou University, Chinese Academy of Sciences, Shanghai Institute of Materia Medica, University of Chinese Academy of Sciences, State Key Laboratory of Drug Research
Language: English

Topic: Cancer-related gene regulation
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: green

Funders: National Natural Science Foundation of China, Natural Science Foundation of Fujian Province, K. C. Wong Education Foundation
Awards: G1334544775, G1498816274, G2221565187, G3350207539, G46207576, G4778903190, G4796892299, G5473757189, G7269206311, G7381190729, G747525406, G7706167721
OpenAlex ID: W3091068616
FWCI: 0.282
Cites: 25
Cited by: 9
Related to: 10
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