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Discovery of novel, potent and orally efficacious inhibitor of neutral amino acid transporter B0AT1 (SLC6A19)

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Year: 2021
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2021.128421
Authors: Jigar Desai, Bhaumin Patel, Brijesh Darji, Archana Gite, Nandini Panchal, Gokul Bhosale, Sandeep Shedage, Sandip Patel, Pravin Kadam, Gautam Patel, Brijesh Kumar Srivastava, Amit Joharapurkar, Samadhan Kshirsagar, Poonam Giri, Hitesh Bhayani, Ankit Patel, Krishnarup Ghoshdastidar, Debdutta Bandyopadhyay, Sanjay Kumar, Mukul Jain, Rajiv Sharma
Institution: Zydus Lifesciences Limited (India)
Language: English

Topic: Amino Acid Enzymes and Metabolism
Subfield: Biochemistry
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W3210376081
FWCI: 1.128
Cites: 21
Cited by: 15
Related to: 10
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