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Mutant‐Selective Allosteric EGFR Degraders are Effective Against a Broad Range of Drug‐Resistant Mutations

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Year: 2020
Type: article
Source: Angewandte Chemie
DOI: 10.1002/ange.202003500
Authors: Jaebong Jang, Ciric To, Dries J. H. De Clercq, Eunyoung Park, Charles M. Ponthier, Bo Hee Shin, Mierzhati Mushajiang, Radosław P. Nowak, Eric S. Fischer, Michael J. Eck, Pasi A. Jänne, Nathanael S. Gray
Institutions: Harvard University, Korea University, Dana-Farber Cancer Institute, Dana-Farber/Harvard Cancer Center
Language: English

Topic: Lung Cancer Treatments and Mutations
Subfield: Pulmonary and Respiratory Medicine
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Institutes of Health, National Cancer Institute
Awards: Protein Kinase Therapeutic Targets for Non-Small Cell Lung Carcinoma, G7768958537, G9000260971
OpenAlex ID: W4213237202
FWCI: 1.475
Cites: 44
Cited by: 16
Related to: 10
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