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Discovery of novel analogs of KHS101 as transforming acidic coiled coil containing protein 3 (TACC3) inhibitors for the treatment of glioblastoma

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Year: 2022
Type: article
Source: European Journal of Medicinal Chemistry
DOI: 10.1016/j.ejmech.2022.114874
Authors: Wenxuan Zhao, Xuyang Sun, Lei Shi, Shi-zhong Cai, Zhou-rui Ma
Institutions: First People's Hospital of Kunshan, Nanjing Medical University, Jiangsu University, Soochow University, Children's Hospital of Suzhou University
Language: English

Topic: Synthesis and biological activity
Subfield: Organic Chemistry
Field: Chemistry
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Jiangsu Commission of Health, National Natural Science Foundation of China
Awards: miR-125b抑制剂增敏脱甲氧基姜黄素和替莫唑胺对胶质瘤干细胞的作用及其机制研究, G3557289753, G3901789764, G5081699786, G6833998682
OpenAlex ID: W4307303928
FWCI: 0.537
Cites: 37
Cited by: 8
Related to: 10
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