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Down‐Regulation of OATP1B1‐Mediated Transport by Mammalian Target of Rapamycin (mTOR) Inhibitors Everolimus and Sirolimus: Potential Mechanism and Implication in OATP‐Mediated Drug‐Drug Interactions

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Year: 2017
Type: article
Source: The FASEB Journal
DOI: 10.1096/fasebj.31.1_supplement.1062.9
Authors: Taleah Farasyn, Sonia Pahwa, Xueying Wang, Pengyue Zhang, Kai Ding, Lang Li, Wei Yue
Institutions: University of Oklahoma, Indiana University Indianapolis, Indiana University School of Medicine
Language: English

Topic: Drug Transport and Resistance Mechanisms
Subfield: Oncology
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: National Institutes of Health, National Institute of General Medical Sciences, National Institute of Diabetes and Digestive and Kidney Diseases, U.S. National Library of Medicine
Awards: G4422131921, Function and regulation of OATP1B1 and OATP1B3, Drug-Drug Interactions Involving Antidiabetic Agents, Evidence-based Drug-Interaction Discovery: In-Vivo, In-Vitro and Clinical
OpenAlex ID: W4389022554
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