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Non-kinase off-target inhibitory activities of clinically-relevant kinase inhibitors

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Year: 2024
Type: review
Source: European Journal of Medicinal Chemistry
DOI: 10.1016/j.ejmech.2024.116540
Authors: Nickolas R. Brauer, Allison L. Kempen, Delmis Hernandez, Herman O. Sintim
Institutions: Purdue University West Lafayette, Purdue University Institute for Cancer Research
Language: English

Topic: Computational Drug Discovery Methods
Subfield: Computational Theory and Mathematics
Field: Computer Science
Domain: Physical Sciences
SDG: Good health and well-being

Open Access status: bronze

Funders: National Institutes of Health, National Cancer Institute
Awards: 3H-pyrazolo[4,3-f]quinoline-containing compounds as selective and tunable protein kinase inhibitors, G7286605037, G9000139669
OpenAlex ID: W4399208050
FWCI: 0.475
Cites: 138
Cited by: 17
Related to: 10
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