Work

Synthesis and evaluation of 3,4,5-trisubstituted triazoles as G protein-biased kappa opioid receptor agonists

Year: 2024

Type: article

Source: European Journal of Medicinal Chemistry

DOI: 10.1016/j.ejmech.2024.116627

Authors: Ashley E. Trojniak, Vuong Q. Dang, Kerri M. Czekner, Robin J. Russo, Lilyan M. Mather, Edward L. Stahl, Michael D. Cameron, Laura M. Bohn, Jeffrey Aubé

Institutions: University of North Carolina at Chapel Hill, The Herbert Wertheim UF Scripps Institute for Biomedical Innovation & Technology

Language: English

Topic: Neuropeptides and Animal Physiology

Subfield: Cellular and Molecular Neuroscience

Field: Neuroscience

Domain: Life Sciences

Open Access status: bronze

Funders: National Institutes of Health, Office of the Director, University of North Carolina at Chapel Hill, National Institute of Mental Health, National Institute on Drug Abuse, NIH Office of the Director, National Cancer Institute, Eshelman Institute for Innovation, University of North Carolina at Chapel Hill

Awards: Biased Kappa Opioid Agonists as Non-addictive Analgesics, G1775929769, G3201181780, Request for a 500 MHz NMR console and nitrogen-cooled cryoprobe, G8691474425, Novel Probes of the Kappa Opioid Receptor: Chemistry, Pharmacology, and Biology, Cancer Center Support Grant

OpenAlex ID: W4400082254

FWCI: 2.141

Cites: 63

Cited by: 13

Related to: 10