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Development and characterization of pyridyl carboxamides as potent and highly selective Nav1.8 inhibitors

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Year: 2024
Type: article
Source: Bioorganic & Medicinal Chemistry Letters
DOI: 10.1016/j.bmcl.2024.130059
Authors: Michael Poslusney, Glen Ernst, Yifang Huang, Aaron C. Gerlach, Mark L. Chapman, Sónia Santos, James C. Barrow
Institutions: Lieber Institute for Brain Development, Duke University Hospital, Johns Hopkins University, Johns Hopkins Medicine
Language: English

Topic: Ion channel regulation and function
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: Lieber Institute for Brain Development
OpenAlex ID: W4405045680
FWCI: 0.407
Cites: 34
Cited by: 3
Related to: 10
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