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MoA Studies of the TEAD P-Site Binding Ligand MSC-4106 and Its Optimization to TEAD1-Selective Amide M3686

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Year: 2024
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.4c01949
Authors: Timo Heinrich, Daniel Schwarz, Carl Petersson, Jakub Gunera, Sakshi Garg, Richard Schneider, Marina Keil, Lisa Grimmeisen, Andrea Unzue Lopez, Lisa Albers, Sarah Schlesiger, Alessia Gambardella, Joerg Bomke, Emma Carswell, Heike Schilke, Patrizia Diehl, Benjamin Doerfel, Djordje Musil, Elisabeth Trivier, Rebecca Broome, Sam Marshall, Alexander Balsiger, Erik Friedrich, Ana R. Lemos, Sandra P. Santos, Pedro M. F. Sousa, Filipe Freire, Tiago M. Bandeiras, Alessio Bortoluzzi, Dirk Wienke
Institutions: Merck Healthcare KGaA, Darmstadt (Germany), Cancer Research Horizons, The Francis Crick Institute, Instituto de Biologia Experimental e Tecnológica
Language: English

Topic: Hippo pathway signaling and YAP/TAZ
Subfield: Cell Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4405641929
FWCI: 1.886
Cites: 32
Cited by: 10
Related to: 10
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