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Discovery of potent free fatty acid receptor 1 full agonists with a novel scaffold bearing conjugated double bond linker

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Year: 2025
Type: article
Source: Bioorganic & Medicinal Chemistry
DOI: 10.1016/j.bmc.2025.118158
Authors: Ziwei Yang, Jun Sun, Tifei Xu, Yu Wang, Jiahui Fang, Kai Wang, Shimeng Guo, Xin Xie, Jianhua Shen
Institutions: Chinese Academy of Sciences, Shanghai Institute of Materia Medica, University of Chinese Academy of Sciences, State Key Laboratory of Drug Research, Tongji University
Language: English

Topic: Diabetes Treatment and Management
Subfield: Endocrinology, Diabetes and Metabolism
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funder: National Natural Science Foundation of China
Awards: G1522379658, G2986465039, G6669830404
OpenAlex ID: W4408434819
FWCI:
Cites: 26
Cited by:
Related to: 10
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