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Abstract 6378: Brain-penetrant molecular glue degraders targeting ALK via a novel degron: a potential therapeutic approach for ALK-positive NSCLC

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Year: 2025
Type: conference-abstract
Source: Cancer Research
DOI: 10.1158/1538-7445.am2025-6378
Authors: Zheng Wang, Massimo Ammirante, Martina Malatesta, Alex Cortez, Young Chen, Jinyi Zhu, Dahlia Weiss, Vijaya Lakshmi Dommeti, Geraldine Hernandez, Joshua M. Baughman, Adwait Sathe, Matthew Groza, Maria Donoso, Roxxana Beltran, Regina Paramitha, Ryan Davison, Atefeh Garzan, Barbra Pagarigan, Michelle Slade, Jacobo Fuentes, Jennifer Buenviaje, Shan Yu, Xinde Zheng, Andres H de la Peña, Mariko Riley, Gabe Mintier, Surendra Nayak, Shuichan Xu, Rama Narla, Ellen Filvaroff, Deborah Mortensen, Lihong Shi, Celia Fontanillo Fontanillo, Christoph Zapf, Neil Bence, Mark Rolfe
Institution: Bristol-Myers Squibb (United States)
Language: English

Topic: Protein Degradation and Inhibitors
Subfield: Molecular Biology
Field: Biochemistry, Genetics and Molecular Biology
Domain: Life Sciences
SDG: Good health and well-being

Open Access status: closed
OpenAlex ID: W4409631536
Cites:
Cited by: 3
Related to: 10
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