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Strategic Design and Optimization of Umifenovir Analogues: Balancing Antiviral Efficacy and hERG Toxicity against SARS-CoV-2

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Year: 2025
Type: article
Source: Journal of Medicinal Chemistry
DOI: 10.1021/acs.jmedchem.4c03093
Authors: Israful Hoque, Nittu Singh, Uddipta Ghosh Dastidar, Alna Kuriyickal Martin, Akshay Joshi, Yogesh Sardana, Ravneet Singh Chawla, Nirmal Das, Binita Patra, Renuga Devi, Satyajeet Das, Dipankar Das, Sahil Kumar, Rajesh P. Ringe, Kiran Kumar Bokara, Krishan Gopal Thakur, Arindam Talukdar
Institutions: Indian Institute of Chemical Biology, Institute of Microbial Technology, Council of Scientific and Industrial Research, Academy of Scientific and Innovative Research, Centre for Cellular and Molecular Biology
Language: English

Topic: SARS-CoV-2 and COVID-19 Research
Subfield: Infectious Diseases
Field: Medicine
Domain: Health Sciences
SDG: Good health and well-being

Open Access status: closed

Funders: Council of Scientific and Industrial Research, India, University Grants Commission
Award: G1276211090
OpenAlex ID: W4409694923
FWCI: 9.92
Cites: 58
Cited by: 14
Related to: 10
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